How to cite this paper
Kshatriya, M & Gajjar, J. (2025). Benzotriazole and its derivatives: A comprehensive review of its synthesis, activities and applications.Current Chemistry Letters, 14(2), 299-322.
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1. Zeng, H., Prato, S., Fasoli, E., Mariani, E., & Tatti, E. (2020). Low temperature magnetic behavior of benzotriazole molecules. Phys. Chem. Chem. Phys., 22, 4200-4207.
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3. Singh, P., & Gu, M. (2021). Electrochemical and surface investigation on benzotriazole-functionalized materials. Electrochim. Acta, 390, 138857.
4. Wang, L., Zhang, Y., & Zhang, X. (2019). Corrosion protection of copper by benzotriazole derivatives. Corros. Sci., 158, 108092.
5. Finsgar, M. (2019). Recent advances in the application of benzotriazole as a corrosion inhibitor. Corros. Eng. Sci. Technol., 54(5), 343-355.
6. Meier, P., & Klinsch, C. (2020). Comprehensive analysis of benzotriazole derivatives in chemical applications. Appl. Sci., 10(11), 3879.
7. Sumran, G.; Jain, N.; Kumar, P.; Aggarwal, R. Trifluoromethyl‐β‐dicarbonyls as versatile synthons in synthesis of heterocycles. Chem. Eur. J. 2024, 30 (11), e202303599.
8. Garg, A.; Bhalla, A. Environmental-benign pathways for the synthesis of medicinally relevant heterocycles. In Green Approaches in Medicinal Chemistry for Sustainable Drug Design; Elsevier, 2024; pp. 361–396.
9. Kushwaha, P.; Rashi; Bhardwaj, A.; Khan, D. Synthetic approaches toward imidazo‐fused heterocycles: a comprehensive review. J. Heterocycl. Chem. 2024.
10. Li, J.; Dong, Z.; Zhao, C. Recent progress for the construction of eight-membered nitrogen-heterocycles. New J. Chem. 2024.
11. Bendi, A.; Yadav, P.; Saini, K.; Singh Bhathiwal, A.; Raghav, N. A comprehensive examination of heterocyclic scaffold chemistry for antitubercular activity. Chem. Biodivers. 2024, e202400067.
12. Beigiazaraghbelagh, P.; Poursattar Marjani, A. Carbon-based catalysts: advances in synthesizing N-heterocyclic compounds using graphene family and graphite oxide. Res. Chem. Intermed. 2024, 50 (2), 485–531.
13. Sadowski, M.; Kula, K. Unexpected course of reaction between (1E, 3E)-1,4-dinitro-1,3-butadiene and N-methyl azomethine ylide—a comprehensive experimental and quantum-chemical study. Molecules 2024, 29 (21), 5066.
14. Sadowski, M.; Dresler, E.; Zawadzińska, K.; Wróblewska, A.; Jasiński, R. Syn-propanethial S-oxide as an available natural building block for the preparation of nitro-functionalized, sulfur-containing five-membered heterocycles: an MEDT study. Molecules 2024, 29 (20), 4892.
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21. Balta, P., & Scott, R. (2018). A review on the electrochemical behavior of benzotriazole. Electrochim. Acta, 289, 243-253.
22. Choudhury, K., & Nandi, A. (2020). Benzotriazole as a corrosion inhibitor in acidic media. Arab. J. Chem., 13(10), 7548-7562.
23. Roy, D., Mukherjee, S., & Das, S. (2019). Electrochemical analysis of benzotriazole-coated metals. J. Chem. Eng., 66(4), 1224-1231.
24. Prabhu, R., & Ananda, S. (2020). Corrosion inhibition and surface protection studies of benzotriazole derivatives. J. Mol. Liq., 310, 113235.
25. Hussein, A., & Haridy, R. (2019). Electrochemical properties of benzotriazole in various pH environments. J. Electrochem. Soc., 166(10), 613-619.
26. Hernandez, M., Torres, T., & Morales, P. (2020). Benzotriazole derivatives as efficient corrosion inhibitors. Corros. Sci., 177, 108928.
27. Reddy, P., & Chandra, A. (2021). Application of benzotriazole in advanced materials. Appl. Sci., 11(2), 387.
28. Li, T., Zhao, Y., & Guo, Z. (2019). Enhanced performance of benzotriazole in corrosive environments. Corros. Eng. Sci. Technol., 54(2), 98-106.
29. Xie, L., Yang, Y., & Zhu, Q. (2018). Chemical and electrochemical insights on benzotriazole coating behavior. J. Phys. Chem. C, 122(14), 7334-7343.
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2. McConville, L., Law, G., & Long, J. (2021). Benzotriazole derivatives in corrosion inhibition: A critical review. Prog. Org. Coat., 158, 106295.
3. Singh, P., & Gu, M. (2021). Electrochemical and surface investigation on benzotriazole-functionalized materials. Electrochim. Acta, 390, 138857.
4. Wang, L., Zhang, Y., & Zhang, X. (2019). Corrosion protection of copper by benzotriazole derivatives. Corros. Sci., 158, 108092.
5. Finsgar, M. (2019). Recent advances in the application of benzotriazole as a corrosion inhibitor. Corros. Eng. Sci. Technol., 54(5), 343-355.
6. Meier, P., & Klinsch, C. (2020). Comprehensive analysis of benzotriazole derivatives in chemical applications. Appl. Sci., 10(11), 3879.
7. Sumran, G.; Jain, N.; Kumar, P.; Aggarwal, R. Trifluoromethyl‐β‐dicarbonyls as versatile synthons in synthesis of heterocycles. Chem. Eur. J. 2024, 30 (11), e202303599.
8. Garg, A.; Bhalla, A. Environmental-benign pathways for the synthesis of medicinally relevant heterocycles. In Green Approaches in Medicinal Chemistry for Sustainable Drug Design; Elsevier, 2024; pp. 361–396.
9. Kushwaha, P.; Rashi; Bhardwaj, A.; Khan, D. Synthetic approaches toward imidazo‐fused heterocycles: a comprehensive review. J. Heterocycl. Chem. 2024.
10. Li, J.; Dong, Z.; Zhao, C. Recent progress for the construction of eight-membered nitrogen-heterocycles. New J. Chem. 2024.
11. Bendi, A.; Yadav, P.; Saini, K.; Singh Bhathiwal, A.; Raghav, N. A comprehensive examination of heterocyclic scaffold chemistry for antitubercular activity. Chem. Biodivers. 2024, e202400067.
12. Beigiazaraghbelagh, P.; Poursattar Marjani, A. Carbon-based catalysts: advances in synthesizing N-heterocyclic compounds using graphene family and graphite oxide. Res. Chem. Intermed. 2024, 50 (2), 485–531.
13. Sadowski, M.; Kula, K. Unexpected course of reaction between (1E, 3E)-1,4-dinitro-1,3-butadiene and N-methyl azomethine ylide—a comprehensive experimental and quantum-chemical study. Molecules 2024, 29 (21), 5066.
14. Sadowski, M.; Dresler, E.; Zawadzińska, K.; Wróblewska, A.; Jasiński, R. Syn-propanethial S-oxide as an available natural building block for the preparation of nitro-functionalized, sulfur-containing five-membered heterocycles: an MEDT study. Molecules 2024, 29 (20), 4892.
15. Aute, D.; Parhad, A.; Vikhe, V.; Uphad, B.; Gadhave, A. Aluminized polyborate catalyzed efficient solvent-free synthesis of 1,8-dioxo-decahydroacridines via Hantzsch condensation. Curr. Chem. Lett. 2024, 13 (2), 417–424.
16. Cho, Y., Kang, M., & Kim, J. (2020). Effects of benzotriazole on copper corrosion in chloride media. Corros. Sci., 173, 108760.
17. Xu, Q., Chen, M., & Ren, Q. (2018). Electrochemical and surface study of benzotriazole films. J. Appl. Electrochem., 48(8), 853-860.
18. Sun, J., Lu, L., & Han, H. (2019). Synthesis and application of benzotriazole-functionalized materials. Chem. Eng. J., 365, 1-10.
19. Yan, W., & Yin, J. (2021). Advanced applications of benzotriazole as a corrosion inhibitor. Appl. Surf. Sci., 563, 150255.
20. Igarashi, M., Saito, R., & Matsumoto, T. (2019). Influence of benzotriazole on the localized corrosion of copper. Electrochim. Acta, 318, 556-562.
21. Balta, P., & Scott, R. (2018). A review on the electrochemical behavior of benzotriazole. Electrochim. Acta, 289, 243-253.
22. Choudhury, K., & Nandi, A. (2020). Benzotriazole as a corrosion inhibitor in acidic media. Arab. J. Chem., 13(10), 7548-7562.
23. Roy, D., Mukherjee, S., & Das, S. (2019). Electrochemical analysis of benzotriazole-coated metals. J. Chem. Eng., 66(4), 1224-1231.
24. Prabhu, R., & Ananda, S. (2020). Corrosion inhibition and surface protection studies of benzotriazole derivatives. J. Mol. Liq., 310, 113235.
25. Hussein, A., & Haridy, R. (2019). Electrochemical properties of benzotriazole in various pH environments. J. Electrochem. Soc., 166(10), 613-619.
26. Hernandez, M., Torres, T., & Morales, P. (2020). Benzotriazole derivatives as efficient corrosion inhibitors. Corros. Sci., 177, 108928.
27. Reddy, P., & Chandra, A. (2021). Application of benzotriazole in advanced materials. Appl. Sci., 11(2), 387.
28. Li, T., Zhao, Y., & Guo, Z. (2019). Enhanced performance of benzotriazole in corrosive environments. Corros. Eng. Sci. Technol., 54(2), 98-106.
29. Xie, L., Yang, Y., & Zhu, Q. (2018). Chemical and electrochemical insights on benzotriazole coating behavior. J. Phys. Chem. C, 122(14), 7334-7343.
30. Kumar, A., Mishra, R., & Sharma, S. (2019). An overview of benzotriazole derivatives for corrosion protection. Prog. Org. Coat., 134, 124-130.
31. Ibon, A., Cossío, F.P., Elguero, J., Fresno, N., Hernandez-Folgado, L., García-Granda, S., Menéndez-Taboada, L., Pérez-Fernández, R., Reviriego, F., & Vázquez-Viñuela, L. (2013). Reaction of NH-indazoles with 1-fluoro-2,4-dinitrobenzene: Unusual formation of benzotriazole-N-oxides. New J. Chem., 37, 1756-1763.
32. Lee, Y.H., Hong, M.S., Ko, S.J., & Kim, J.G. (2021). Effect of benzotriazole on localized corrosion of copper. Materials, 14(11), 2722.
33. Liu, L., Shuang, L., Qi, Y., Wu, X., & Xie, J. (2020). Corrosion inhibition behavior of benzotriazole derivatives on copper. Anti-Corros. Methods Mater., 67(4), 123-129.
34. Youssef, Y.M., Ahmed, N.M., Nosier, S.A., Farag, H.A., & Abdel-Aziz, M.H. (2020). Utilizing benzotriazole for corrosion protection in metals under flow conditions. Chem. Pap., 74(8), 3395-3408.
35. Paoletti, N., & Supuran, C.T. (2024). Benzothiazole derivatives in antitumor agents. Arch. Pharm., 357(6), e200059.
36. Ibba, R., Piras, S., Corona, P., Riu, F., Loddo, R., Delogu, I., Collu, G., Sanna, G., Caria, P., Dettori, T., & Carta, A. (2021). Synthesis, antitumor, and antiviral activities of new benzotriazole-dicarboxamide derivatives. Front. Chem., 9, 660424.
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