How to cite this paper
Agrawal, N. (2021). Synthetic and therapeutic potential of 4-thiazolidinone and its analogs.Current Chemistry Letters, 10(2), 119-138.
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3. Mishchenko M., Shtrygol S., Kaminskyy D., Lesyk R. (2020) Thiazole-bearing 4-thiazolidinones as new anticonvulsant agents. Sci. Pharm., 88 (1), 16-30.
4. Ekinci A. S., Moncol J., Krishna V S., Sriram D., Özadali-Sari K. (2020) 5-Methyl-4-thiazolidinones, Synthesis and evaluation as antitubercular agents. J. Res. Pharm., 24 (1), 30–37.
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6. Güzeldemirci N. U., Pehlivan E., Naesens L. (2018) Synthesis and antiviral activity evaluation of new 4-thiazolidinones bearing an imidazo2,1-b.thiazole moiety. Marmara Pharm. J., 22 (2), 237–248.
7. Gomathy S., Singh G., Gowramma B. Antony A. S., Elango K. (2012) Synthesis and anti-Parkinson′s screening of some novel 2-(naphthalen-1-yl)-N-2-substituted (4-oxothiazolidin-3-yl).acetamide derivatives. Int. J. Heal. Allied Sci.,1 (4), 244-248.
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9. Anekal D. P., Biradar J. S. (2017) Synthesis and biological evaluation of novel Indolyl 4-thiazolidinones bearing thiadiazine nucleus. Arab. J. Chem., 10 (suppl 2), S2098–S2105.
10. Shinde R. S., Masand V. H., Patil M. K. (2019) Antiinflammatory activity of triazine thiazolidinone derivatives, molecular docking and pharmacophore modeling. Indian J. Pharm. Sci., 81 (5), 851–858.
11. Incerti M., Crascì L., Vicini P., Aki E., Yalcin I., Ertan-Bolelli T., et al. (2018) 4-thiazolidinone derivatives as MMP inhibitors in tissue damage: Synthesis, biological evaluation and docking studies. Molecules, 23 (2), 1–18.
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15. Rocha-Roa C., Molina D., Cardona N. (2018) A perspective on thiazolidinone scaffold development as a new therapeutic strategy for Toxoplasmosis. Front. Cell Infect. Microbiol., 8, 360-368.
16. Devinyak O., Zimenkovsky B., Lesyk R. (2013) Biologically active 4-thiazolidinones, a review of QSAR studies and QSAR modeling of antitumor activity. Curr. Top. Med. Chem.,12 (24), 2763–2784.
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29. Nampurath G. K., Mathew S. P., Khanna V., Zachariah R. T., Kanji S., Chamallamudi M. R. (2008) Assessment of hypolipidaemic activity of three thiazolidin-4-ones in mice given high-fat diet and fructose. Chem. Biol. Interact., 171 (3), 363–368.
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2. Cheddie A., Shintre S. A., Bantho A., Mocktar C., Koorbanally N. A. (2020) Synthesis and antibacterial activity of a series of 2-trifluoromethylbenzimidazole-thiazolidinone derivatives. J. Heterocycl. Chem., 57 (1), 299–307.
3. Mishchenko M., Shtrygol S., Kaminskyy D., Lesyk R. (2020) Thiazole-bearing 4-thiazolidinones as new anticonvulsant agents. Sci. Pharm., 88 (1), 16-30.
4. Ekinci A. S., Moncol J., Krishna V S., Sriram D., Özadali-Sari K. (2020) 5-Methyl-4-thiazolidinones, Synthesis and evaluation as antitubercular agents. J. Res. Pharm., 24 (1), 30–37.
5. Gawrońska-Grzywacz M., Popiołek Ł, Natorska-Chomicka D., Piątkowska-Chmiel I., Izdebska M., Herbet M., et al. (2019) Novel 2,3-disubstituted 1,3-thiazolidin-4-one derivatives as potential antitumor agents in renal cell adenocarcinoma. Oncol. Rep., 41 (1), 693–701.
6. Güzeldemirci N. U., Pehlivan E., Naesens L. (2018) Synthesis and antiviral activity evaluation of new 4-thiazolidinones bearing an imidazo2,1-b.thiazole moiety. Marmara Pharm. J., 22 (2), 237–248.
7. Gomathy S., Singh G., Gowramma B. Antony A. S., Elango K. (2012) Synthesis and anti-Parkinson′s screening of some novel 2-(naphthalen-1-yl)-N-2-substituted (4-oxothiazolidin-3-yl).acetamide derivatives. Int. J. Heal. Allied Sci.,1 (4), 244-248.
8. Panico A. M., Vicini P., Geronikaki A., Incerti M., Cardile V., Crascì L., et al. (2011) Heteroarylimino-4-thiazolidinones as inhibitors of cartilage degradation. Bioorg. Chem., 39 (1), 48–52.
9. Anekal D. P., Biradar J. S. (2017) Synthesis and biological evaluation of novel Indolyl 4-thiazolidinones bearing thiadiazine nucleus. Arab. J. Chem., 10 (suppl 2), S2098–S2105.
10. Shinde R. S., Masand V. H., Patil M. K. (2019) Antiinflammatory activity of triazine thiazolidinone derivatives, molecular docking and pharmacophore modeling. Indian J. Pharm. Sci., 81 (5), 851–858.
11. Incerti M., Crascì L., Vicini P., Aki E., Yalcin I., Ertan-Bolelli T., et al. (2018) 4-thiazolidinone derivatives as MMP inhibitors in tissue damage: Synthesis, biological evaluation and docking studies. Molecules, 23 (2), 1–18.
12. Bonn G. F., Otrzonsek G., Windsheimer F, Schneider B. (1980) Long-term antihypertensive therapy with Etozoline. Med. Welt., 31 (16), 603–607.
13. Ramirez M. A., Borja N. L. (2008) Epalrestat, An aldose reductase inhibitor for the treatment of diabetic neuropathy. Pharmacotherapy, 28 (5), 646–655.
14. Nirwan S., Chahal V., Kakkar R. (2019) Thiazolidinones, synthesis, reactivity, and their biological applications. J. Heterocycl. Chem., 56 (4), 1239–1253.
15. Rocha-Roa C., Molina D., Cardona N. (2018) A perspective on thiazolidinone scaffold development as a new therapeutic strategy for Toxoplasmosis. Front. Cell Infect. Microbiol., 8, 360-368.
16. Devinyak O., Zimenkovsky B., Lesyk R. (2013) Biologically active 4-thiazolidinones, a review of QSAR studies and QSAR modeling of antitumor activity. Curr. Top. Med. Chem.,12 (24), 2763–2784.
17. Jain A. K., Vaidya A., Ravichandran V., Kashaw S. K., Agrawal R. K. (2012) Recent developments and biological activities of thiazolidinone derivatives: A review. Bioorg. Med. Chem., 20 (11), 3378–3395.
18. Hamama W. S., Ismail M. A., Shaaban S., Zoorob H. H. (2008) Progress in the chemistry of 4- thiazolidinones. J. Heterocycl. Chem., 45 (4), 939–956.
19. Kumar A., Rajput C. S., Bhati S. K. (2007) Synthesis of 3-4′-(p-chlorophenyl)-thiazol-2′-yl.-2-(substituted azetidinone/thiazolidinone)-aminomethyl.-6-bromoquinazolin-4-ones as anti-inflammatory agent. Bioorg. Med. Chem., 15 (8), 3089–3096.
20. Sharma R. C., Kumar D. (2000) Synthesis of some new thiazolidin-4-ones as possible antimicrobial agents. J. Indian Chem. Soc., 77, 492–493.
21. Ojha S., Ameta U., Dhakar N., Talesara G. L. (2007) Synthesis and characterization of some alkoxypathalimide derivatives of benzotriazolythiadiazoles and benzotriazolyl thiazolidinones. Indian J. Chem.-Sect. B Org. Med. Chem., 46 (5), 860–865.
22. Vicini P., Geronikaki A., Incerti M., Zani F., Dearden J., Hewitt M. (2008) 2-heteroarylimino-5-benzylidene-4-thiazolidinones analogues of 2-thiazolylimino-5-benzylidene-4-thiazolidinones with antimicrobial activity: Synthesis and structure–activity relationship. Bioorg. Med. Chem., 16 (7), 3714–3724.
23. Ottanà R., Maccari R., Giglio M., Del Corso A., Cappiello M., Mura U., et al. (2011) Identification of 5-arylidene-4-thiazolidinone derivatives endowed with dual activity as aldose reductase inhibitors and antioxidant agents for the treatment of diabetic complications. Eur. J. Med. Chem., 46 (7), 2797–2806.
24. Verma P., Kamboj V. (2010) Synthesis and antidiabetic activity of N’-3-(alkyl/aryl substituted)-4-oxo-1,3 thiazolidin-2-yleidene.-2-(pyrazin-2-yloxy)acetohydrazide. Acta Pharm. Sci., 52 (4), 411–415.
25. Sharma P., Shrivastava B., Lamba H S., Sharma J., Sharma L. (2010) Synthesis and pharmacological study of 4-thiazolidinone derivatives. Int. J. Compr. Pharm., 3, 1-6.
26. Firke S. D., Firake B. M., Chaudhari R. Y., Patil V. R. (2009) Synthetic and pharmacological evaluation of some pyridine containing thiazolidinones. Asian J. Res. Chem., 2 (2), 157–160.
27. Imran M., Yar M. S., Khan S. A. (2009) Synthesis and antihyperglycemic activity of 2-(substituted phenyl)-3-{4-(1-naphthyl)-1,3-thiazol-2-yl-amino}-4-oxo-1,3-thiazolidin-5-ylacetic acid derivatives. Acta Pol. Pharm.-Drug Res., 66 (1), 51–56.
28. Kishore A., Nampurath G. K., Mathew S. P., Zachariah R. T., Potu B. K., Rao M. S., et al. (2009) Antidiabetic effect through islet cell protection in streptozotocin diabetes, A preliminary assessment of two thiazolidin-4-ones in Swiss albino mice. Chem. Biol. Interact., 177 (3), 242–246.
29. Nampurath G. K., Mathew S. P., Khanna V., Zachariah R. T., Kanji S., Chamallamudi M. R. (2008) Assessment of hypolipidaemic activity of three thiazolidin-4-ones in mice given high-fat diet and fructose. Chem. Biol. Interact., 171 (3), 363–368.
30. Singh T., Soni B. K., Reddy B. B.. (2011) Synthesis and evaluation of thiazolidinones derivatives for their pharmacological activity. Int. J. Res. Pharm. Biomed. Sci., 2, 1562–1567.
31. Deep A., Jain S., Sharma P. C. (2010) Synthesis and anti-inflammatory activity of some novel biphenyl-4- carboxylic acid 5-(arylidene)-2-(aryl)-4-oxothiazolidin-3-yl amides. Acta Pol. Pharm.-Drug Res., 67 (1), 63–6 7.
32. Barros C. D., Amato A. A., Oliveira T. B. de, Iannini K. B. R., Silva A. L. da, Silva T. G. da, et al. (2010) Synthesis and anti-inflammatory activity of new arylidene-thiazolidine-2,4-diones as PPARγ ligands. Bioorg. Med. Chem., 18 (11), 3805–3811.
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